Lets Forget AR
10-12-2005, 11:02 PM
Falsodex
(Originally posted on www.*****************.com (http://www.*****************.com/))
Falsodex is an estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) receptor antagonist, which has no agonist effects at all. What it does is downregulates Estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) Receptors (kinda like how Clen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=45) DownRegulates your beta receptors....so you get decreased effects from the stuff). Basically, it binds to the Estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) Receptor more strongly then Tamoxifen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=43), but still has no estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) agonist effects. Here's the interesting part:
The resultant downregulation of your Estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) Receptors from the use of Falsodex results in decreased expression of the Progesterone Receptor as well! Tamoxifen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=43), as we all know, can increase the sides from progesteronic drugs because of an increase in progesterone receptor expression. So you can take this stuff as both an anti-estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) and an anti-progestin! No more buying Arimidex (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=98) or whatever, and Bromocriptine! Sweet, huh?
But here's the part that really gave me a hard-on:
The stuff is administered via an IM injection of 250mgs once per month! And at that dose, it has have most if not all of the same estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) lowering effects of 1mg/day of Arim or 2.5mgs per day of Letrozole (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42), but has the added benefits of lowering progesterone receptor expression.
Enjoy, Kiddies...
References:
(Br J Cancer. 2004 Mar;90 Suppl 1:S15-8)
(Drugs. 2004;64(6):633-48.)
(J Steroid Biochem Mol Biol. 2001 Dec;79(1-5):209-12)
(Originally posted on www.*****************.com (http://www.*****************.com/))
Falsodex is an estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) receptor antagonist, which has no agonist effects at all. What it does is downregulates Estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) Receptors (kinda like how Clen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=45) DownRegulates your beta receptors....so you get decreased effects from the stuff). Basically, it binds to the Estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) Receptor more strongly then Tamoxifen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=43), but still has no estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) agonist effects. Here's the interesting part:
The resultant downregulation of your Estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) Receptors from the use of Falsodex results in decreased expression of the Progesterone Receptor as well! Tamoxifen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=43), as we all know, can increase the sides from progesteronic drugs because of an increase in progesterone receptor expression. So you can take this stuff as both an anti-estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) and an anti-progestin! No more buying Arimidex (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=98) or whatever, and Bromocriptine! Sweet, huh?
But here's the part that really gave me a hard-on:
The stuff is administered via an IM injection of 250mgs once per month! And at that dose, it has have most if not all of the same estrogen (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42) lowering effects of 1mg/day of Arim or 2.5mgs per day of Letrozole (http://www.anabolicreview-research.com/shop/product_info.php?cPath=23&products_id=42), but has the added benefits of lowering progesterone receptor expression.
Enjoy, Kiddies...
References:
(Br J Cancer. 2004 Mar;90 Suppl 1:S15-8)
(Drugs. 2004;64(6):633-48.)
(J Steroid Biochem Mol Biol. 2001 Dec;79(1-5):209-12)